azatadine (optimine) Report issue

Small molecule Approved FDA
ChEMBL DrugBank Drug Central Drugs@FDA KEGG MeSH PubChem repoDB

Active Ingredient History

NOW
  • Now
Azatadine is an antihistamine, which blocks the effects of the naturally occurring chemical histamine in the body. Azatadine is used to treat sneezing; runny nose; itching, watery eyes; hives; rashes; and other symptoms of allergies and the common cold. The antihistamines antagonize those pharmacological effects of histamine, which are mediated through activation of H1- receptor sites and thereby reduce the intensity of allergic reactions and tissue injury response involving histamine release.   NCATS

Chemistry

  • SMILES: CN1CCC(=C2c3ccccc3CCc3cccnc32)CC1
  • InChIKey: SEBMTIQKRHYNIT-UHFFFAOYSA-N
  • Mol. Mass: 290.41
  • ALogP: 3.71
  • ChEMBL Molecules:
    azatadine  
    azatadine maleate  
More Chemistry

Pharmacology

  • Mechanism of Action:
  • Multi-specific: Missing data
  • Black Box: No
  • Availability: Discontinued
  • Delivery Methods: Oral
  • Pro Drug: No

Combination drugs

( azatadine (optimine), pseudoephedrine (Benylin) )

Alternative names

11-(1-methyl-4-piperidinylidene)-6,11-dihydro-5h-benzo[5,6]cyclohepta[1,2-b]pyridine | 6,11-dihydro-11-(1-methyl-4-piperidylidene)-5h-benzo(5,6)cyclohepta(1,2-b)pyridine | azatadin | azatadina | azatadine | azatadine maleate | azatadinum | azatidine | idulamine | idulian | juste brand of azatadine maleate | key brand of azatadine maleate | lergocil | optimine | sch-10649 | schering brand of azatadine maleate | schering-plough brand of azatadine maleate | trinalin | zadine

Organizations (2)

Research & Development (0)

Organization Org Type FDA approvals Clinical Trials involvement Org ID Force Sort

Marketing (2)

Organization Org Type FDA approvals Clinical Trials involvement Org ID Force Sort

Indications (4)

Approved Indications (4)


 

Diaper Rash (approved 1977)

Pruritus (approved 1977)

Sneezing (approved 1977)

Urticaria (approved 1977)

Experimental Indications - Clinical Trial Phases 1-4 (0)

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