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Momelotinib (INN, formerly GS-0387, CYT-387) is an inhibitor of Janus kinases JAK1 and JAK2, acting as an ATP competitor with IC50 values of 11 and 18 nM, respectively. The inhibitor is significantly less active towards other kinases, including JAK3 (IC50 = 0.16 μM).   Wikipedia

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cyt-11387 | cyt387 | cyt 387 | cyt-387 | gs-0387 | momelotinib | momelotinib dihydrochloride

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