cinchocaine (nupercaine) Report issue

Small molecule Approved FDA
ChEMBL DrugBank Drug Central Drugs@FDA KEGG MeSH PubChem repoDB

Active Ingredient History

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Dibucaine is used as a local anesthetic for surface anesthesia. It is one of the most potent and toxic of the long-acting local anesthetics and its parenteral use is restricted to spinal anesthesia. Dibucaine is used to temporarily relieve pain and itching due to: hemorrhoids or other anorectal disorders, sunburn, minor burns, minor cuts; scrapes, insect bites, minor skin irritation. This drug acts via blocking of nerve impulses by decreasing the neuronal membrane's permeability to sodium ions through sodium channel blocking. This reversibly stabilizes the membrane and inhibits depolarization, resulting in the failure of a propagated action potential and subsequent conduction blockade.   NCATS

Chemistry

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Pharmacology

Drug Pricing (per unit)

United States

$0.1442 - $0.1443
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Note: This drug pricing data is preliminary, incomplete, and may contain errors.

Alternative names

2-butoxy-n-[2-(diethylamino)ethyl]-4-quinolinecarboxamide | 2-butoxy-n-(2-(diethylamino)ethyl)cinchoninamide | 2-butoxy-n-(alpha-diethylaminoethyl)cinchoninamide | 2-butoxy-n-(beta-diethylaminoethyl)cinchoninamide | 2-butoxy-quinoline-4-carboxylic acid (2-diethylamino-ethyl)-amide | 2-butoxyquinoline-4-carboxylic acid diethylaminoethylamide | 2-n-butoxy-n-(2-diethylaminoethyl)cinchoninamide | alpha-butyloxycinchonic acid-gamma-diethylethylenediamine | alpha-butyloxycinchoninic acid diethylethylenediamide | cincaine chloride | cinchocaine | cinchocaine hcl | cinchocainum | cincocainio | dermacaine | dibucaine | dibucaine base | dibucaine hcl | dibucaine hydrochloride | heavy solution nupercaine | n-(2-(diethylamino)ethyl)-2-butoxycinchoninamide | nupercainal | nupercaine | percamine

Organizations (2)

Research & Development (0)

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Marketing (2)

Organization Org Type FDA approvals Clinical Trials involvement Org ID Force Sort

Indications (3)

Approved Indications (3)


 

Hemorrhoids

Pain

Sunburn

Experimental Indications - Clinical Trial Phases 1-4 (0)

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