bilastine Report issue

Small molecule Experimental
AACT ChEMBL DrugBank Drug Central KEGG PubChem repoDB

Active Ingredient History

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  • Now
Bilastine is an antihistamine medication used to treat hives (urticaria), allergic rhinitis and itchy inflamed eyes (allergic conjunctivitis) caused by an allergy. It is a second-generation antihistamine and takes effect by selectively inhibiting the histamine H1 receptor, preventing these allergic reactions. Bilastine has an effectiveness similar to cetirizine, fexofenadine, and desloratadine.   Wikipedia

Chemistry

  • SMILES: CCOCCn1c(C2CCN(CCc3ccc(C(C)(C)C(=O)O)cc3)CC2)nc2ccccc21
  • InChIKey: ACCMWZWAEFYUGZ-UHFFFAOYSA-N
  • Mol. Mass: 463.62
  • ALogP: 4.86
  • ChEMBL Molecule:
    bilastine  
More Chemistry

Pharmacology

Alternative names

bellozal | bilastine | bilaxten | f-96221-bm1 | ilaxten

Organizations (32)

Research & Development (32)

Organization Org Type FDA approvals Clinical Trials involvement Org ID Force Sort

Marketing (0)

Organization Org Type FDA approvals Clinical Trials involvement Org ID Force Sort

Indications (11)

Approved Indications (1)


 

Hypersensitivity

Experimental Indications - Clinical Trial Phases 1-4 (11)


 

Asthma (Phase 4)

Chronic Urticaria (Phase 3)

Conjunctivitis (Phase 4)

Conjunctivitis, Allergic (Phase 3)

Healthy Volunteers (Phase 1)

Hypersensitivity (Phase 2)

Pharmacokinetics (Phase 1)

Rhinitis, Allergic (Phase 4)

Rhinitis, Allergic, Perennial (Phase 3)

Rhinitis, Allergic, Seasonal (Phase 4)

Urticaria (Phase 4)

Overview

  • Highest Phase: Phase 4
  • # of Trials: 24
  • # of Trial Organizations: 32

Trials by Phase

Trial Phase Start Date Organizations Indications

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