Pharmacokinetics D010599

Phenomena and Processes [G] » Metabolism [G03] » Pharmacokinetics

Phenomena and Processes [G] » Physiological Phenomena [G07] » Pharmacological and Toxicological Phenomena » Pharmacokinetics

Description

Dynamic and kinetic mechanisms of exogenous chemical DRUG LIBERATION; ABSORPTION; BIOLOGICAL TRANSPORT; TISSUE DISTRIBUTION; BIOTRANSFORMATION; elimination; and DRUG TOXICITY as a function of dosage, and rate of METABOLISM. LADMER, ADME and ADMET are abbreviations for liberation, absorption, distribution, metabolism, elimination, and toxicology.   MeSH

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Subtype Terms (10)

Absorption
11 drugs (4 approved, 7 experimental)

Area Under Curve
3 approved drugs

Biological Availability
104 drugs (71 approved, 33 experimental)

Biotransformation
 

Therapeutic Equivalency
135 drugs (108 approved, 27 experimental)

Tissue Distribution
 


Phase 4 Indicated Drugs (87)

Phase 1 Indicated Drugs (351)

ciprofloxacin (cipro)

clarithromycin (biaxin)

clonazepam (klonopin)

cobicistat (stribild)

cocaine (Erythroxyline)

crd-740

curcumin

d961

dabigatran (pradaxa)

darexaban

darolutamide (Nubeqa)

darunavir (prezista)

dasatinib (sprycel)

dehydroepiandrosterone

denosumab (prolia)

desipramine (pertofrane)

dexmecamylamine

dextromethorphan (delsym)

diclofenac (voltaren)

dienogest (natazia)

digoxin (lanoxin)

dihydroartemisinin

diltiazem (cardizem)

diphencyprone

dofetilide (tikosyn)

ds-1971

ds-8500a

dtri-031

edaravone (radicava)

efavirenz (sustiva)

eflapegrastim (Rolvedon)

enalapril (vasotec)

enclomiphene

endostatin (endostar)

entacapone (comtan)

entospletinib

enzalutamide (xtandi)

Enzaplatovir

Epimedium

erythromycin (ilosone)

esk-001

esomeprazole (nexium)

estetrol (NEXTSTELLIS)

ethinyl estradiol (Estinyl)

etravirine (intelence)

everolimus (zortress)

evolocumab (repatha)

ezetimibe (zetia)

f573

fasiglifam

faxeladol

fenofibrate (fenoglide)

fexofenadine (allegra)

fidaxomicin (dificid)

Filgrastim (neupogen)

fimasartan (kanarb)

finafloxacin (xtoro)

finerenone (KERENDIA)

fludrocortisone (florinef)

fluorescein

Flupirtine (katadolon)

fluvoxamine (luvox)

folic acid

follitropin alfa (Gonal-F)

fostamatinib

fremanezumab (Ajovy)

funapide

furosemide (lasix)

gadopiclenol (Elucirem)

galantamine (reminyl)

gb1211

ge200486

gemfibrozil (lopid)

gft505

gilteritinib

glimepiride (amaryl)

glycopyrronium (robinul)

gst-hg121

hexyl 5-aminolevulinate (Cysview)

htl0018318

hutrukin

hydrochlorothiazide (esidrix)

hydrocodone (hycodan)

hydronidone

hydroxyzine (vistaril)

Iberdomide

Ibrexafungerp (Brexafemme)

icosapent ethyl (vascepa)

ilaprazole (noltec)

imagabalin

inv-101

ipg7236

ipragliflozin (sublet)

isavuconazium

isavuconazonium (cresemba)

isosorbide (isordil)

jnj-26483327

jnj-42165279

ketoconazole (nizoral)

ketoprofen (orudis)

ketorolac (acuvail)

kt07

lactose

lanifibranor

lansoprazole (prevacid)

laquinimod

levodopa (larodopa)

levofloxacin (levaquin)

levothyroxine (Synthroid)

linaclotide (linzess)

linaprazan

linsitinib

Lisaftoclax

lomitapide (juxtapid)

lopinavir (Kaletra)

loteprednol (lotemax)

lurasidone (latuda)

ly2428703

maraviroc (selzentry)

medicinal charcoal

megestrol (megace)

meloxicam (mobic)

memantine (namenda)

mepolizumab (Nucala)

mesna (mesnex)

methylphenidate (ritalin)

metoprolol (lopressor)

mexiletine (mexitil)

miglitol (glyset)

minocycline (minocin)

mitiglinide (Glufast)

Mizacorat

mk-1064

mk-2048

mk-5890

mk-7252

mln3126

moon kratom yellow

mycophenolate (CellCept)

nafamostat (ronastat)

nalmefene (revex)

naloxone (narcan)

naltrexone (revia)

napabucasin

naproxen (naprosyn)

natrunix

nicergoline (Sermion)

nicotinamide

nicotine (nicorette)

nirmatrelvir (Paxlovid)

norethindrone

norgestimate

norgestrel (Ovral)

noristerat

npc-22

olanzapine (zyprexa)

olokizumab

omalizumab (xolair)

omega-3-carboxylic acids (epanova)

omeprazole (prilosec)

Opigolix

oxymetazoline (ocuclear)

paclitaxel (taxol)

padsevonil

pantoprazole (protonix)

peficitinib (Vonjo)

peginterferon beta-1a (Plegridy)

pemetrexed (alimta)

pertuzumab (perjeta)

pf-00258210

pf-05212372

pioglitazone (actos)

ponesimod (Ponvory)

prasugrel (effient)

pravastatin (pravachol)

prednisone (meticorten)

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