Carfentanil Report issue

Small molecule Experimental
AACT DrugBank MeSH PubChem

Active Ingredient History

NOW
  • Now
Carfentanil or carfentanyl, sold under the brand name Wildnil, is an extremely potent opioid analgesic used in veterinary medicine to anesthetize large animals such as elephants and rhinoceroses. It is typically administered in this context by tranquilizer dart. Carfentanil has also been used in humans to image opioid receptors. It has additionally been used as a recreational drug, typically by injection, insufflation, or inhalation. Deaths have been reported in association with carfentanil.   Wikipedia

Chemistry

  • SMILES: CCC(=O)N(c1ccccc1)C1(C(=O)O[11CH3])CCN(CCc2ccccc2)CC1
  • InChIKey: YDSDEBIZUNNPOB-JVVVGQRLSA-N
  • Mol. Mass: 393.52
  • ALogP: 3.68
  • ChEMBL Molecules:
    [11c]-carfentanil  
    carfentanil  
More Chemistry

Pharmacology

Alternative names

11c-carfentanil | (4-methoxycarbonyl)fentanyl | 4-methoxycarbonylfentanyl | 4-methoxycarbonyl fentanyl | 4-piperidinecarboxylic acid, 4-((1-oxopropyl)phenylamino)-1-(2-phenylethyl)-, methyl ester, 2-hydroxy-1,2,3-propanetricarboxylate (1:1) | carfentanil | carfentanil citrate | carfentanil, (+-)-isomer | carfentanil oxalate | carfentanyl | r31833 | r 31833 | r-31833 | r 33799

Organizations (7)

Research & Development (7)

Organization Org Type FDA approvals Clinical Trials involvement Org ID Force Sort

Marketing (0)

Organization Org Type FDA approvals Clinical Trials involvement Org ID Force Sort

Indications (4)

Approved Indications (0)

Experimental Indications - Clinical Trial Phases 1-4 (4)


 

Healthy Volunteers (Phase 1)

Neuralgia (Phase 2)

Opioid-Related Disorders (Phase 1)

Substance Abuse, Oral (Phase 1)

Overview

  • Highest Phase: Phase 2
  • # of Trials: 4
  • # of Trial Organizations: 7

Trials by Phase

Trial Phase Start Date Organizations Indications

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